Simvastatin

Simvastatin

Lipid-lowering Prescription only ATC code: C10AA01

What it is

Simvastatin is a statin that inhibits HMG-CoA reductase, the enzyme governing cholesterol synthesis in the liver, prompting the liver to clear more LDL cholesterol from the blood. It is used to lower cholesterol, with LDL and total cholesterol tracking the response.

Typical dose
10–40 mg
1× a day
Times
Any time
Evening

Used for

  • Cholesterol

What to know while taking it

It suits evening dosing and can be taken with or without food, but grapefruit is avoided: it blocks the enzyme that breaks simvastatin down, so blood levels climb and with them the risk of muscle damage. The same mechanism rules out clarithromycin and itraconazole, and amlodipine raises levels enough to warrant caution. ALT is monitored for liver strain, and creatine kinase is the test used when muscle symptoms suggest myopathy; the drug also depletes coenzyme Q10. It is not used in pregnancy, since cholesterol is essential to fetal development.

When to see a doctor

Unexplained muscle pain, tenderness or weakness, particularly alongside dark urine or fever, should be assessed by a doctor without delay, as should jaundice, dark urine with abdominal pain, or unusual tiredness. Pregnancy, planned or confirmed, is a reason to see a doctor rather than stopping or continuing alone.

Worth knowing

  • Avoid grapefruit
  • Report unexplained muscle pain
  • Watch liver enzymes
  • Not during pregnancy

Do not combine with

Interacts with

Markers to watch

Nutrients affected

  • coq10 — depleted by

Reference information, not medical advice. Discuss any change with your doctor.